N-[2--[4-[N-(Hexyloxycarbonyl))amidino]phenylaminomethyl]-1-methyl-1H-benzimidazol-5-ylcarbonyl]-N-(2-pyridyl)-beta-alanine ethyl ester CAS: 211915-06 -9
Nomoro ea lethathamo | XD93359 |
Lebitso la Sehlahiswa | N-[2-[4-[N-(Hexyloxycarbonyl))amidino]phenylaminomethyl]-1-methyl-1H-benzimidazol-5-ylcarbonyl]-N-(2-pyridyl)-beta-alanine ethyl ester |
CAS | 211915-06-9 |
Foromo ea molek'hulela | C34H41N7O5 |
Boima ba Molek'hule | 627.73 |
Lintlha tsa polokelo | Ambient |
Tlhaloso ea Sehlahisoa
Ponahalo | Phofo e tšoeu |
Assay | 99% mets |
N-[2-[4-[N-(Hexyloxycarbonyl))amidino]phenylaminomethyl]-1-methyl-1H-benzimidazol-5-ylcarbonyl]-N-(2-pyridyl)-beta-alanine ethyl ester, eo hape e bitsoang motsoako, ke lik'hemik'hale tse rarahaneng le tse khethehileng tse nang le lik'hemik'hale tse ka sebelisoang mafapheng a sa tšoaneng, ho kenyeletsoa k'hemistri ea meriana le nts'etsopele ea lithethefatsi.Nngoe e ka sebelisoang ea motsoako ona ke ts'ebeliso ea eona e le setsi sa meriana.E na le lihlopha tse 'maloa tse sebetsang tse ka fetoloang ho ntlafatsa thepa ea eona ea bongaka.Sebopeho sa motsoako se kenyelletsa reng ea benzimidazole, e tsejoang ka ho bonts'a mesebetsi e fapaneng ea likokoana-hloko.Sena se etsa hore e be sepheo se khahlang bakeng sa lipatlisiso tse ling tsa k'hemistri ea bongaka.Bafuputsi ba ka batlisisa liphello tsa eona tsa phekolo tse ka 'nang tsa e-ba teng, tse kang antimicrobial, anticancer, kapa anti-inflammatory properties.E ka sebetsa e le qalo ea tlhahiso ea lithethefatsi tse ncha kapa motsoako oa metsoako e amanang le sebopeho ka katleho e ntlafetseng le litla-morao tse fokotsehileng.Kopo e 'ngoe ea motsoako e itšetlehile ka tšebeliso ea eona e ka sebelisoang e le sesebelisoa sa lik'hemik'hale lipatlisisong tsa likokoana-hloko.Sebopeho sa eona se ikhethang le lihlopha tse sebetsang li etsa hore e tšoanelehe bakeng sa ho ithuta litšebelisano tsa limolek'hule le mekhoa ea likokoana-hloko.Bafuputsi ba ka sebelisa motsoako ho batlisisa sepheo kapa litsela tse itseng liseleng le linthong tse phelang.Ka ho kenyelletsa motsoako litekong, bo-rasaense ba ka fumana kutloisiso e ntle ea mekhoa ea mafu a itseng kapa mekhoa ea 'mele.Tsebo ena e ka kenya letsoho ho nts'etsopele ea mekhoa e mecha ea phekolo kapa ho khetholla lipakane tse ncha tsa lithethefatsi.Ho feta moo, motsoako o ka sebelisoa e le mohaho oa ho haha motsoako oa manyolo.Sebopeho sa eona se rarahaneng se fana ka sethala se setle sa ho theha limolek'hule tse rarahaneng tse nang le thepa e hlophisitsoeng.Litsebi tsa lik'hemik'hale tsa 'mele li ka fetola lihlopha tse sebetsang tsa motsoako ho hlahisa lihlahisoa tse nang le lik'hemik'hale tse khethehileng kapa tsa likokoana-hloko.Ts'ebetso ena e fapaneng e lumella ho kopanngoa ha metsoako e ka sebelisoang lits'ebetsong tse fapaneng, ho kenyelletsa le mahlale a lisebelisoa, lipatlisiso tsa limolek'hule, kapa lithuto tsa biology ea lik'hemik'hale. katleho.Lithuto tse felletseng, ho kenyeletsoa litlhahlobo tsa pharmacokinetic, litlhahlobo tsa chefo, le litlhahlobo tse qaqileng tsa baeloji, li bohlokoa ho fumana hore na e sebetsa joang joalo ka moemeli oa lithethefatsi kapa joalo ka sesebelisoa sa lik'hemik'hale se sebetsang.Ho feta moo, liprothokholo le litataiso tsa ts'ireletso li tlameha ho lateloa ka thata ha ho sebetsa le motsoako ho netefatsa boiketlo ba bafuputsi le ho thibela likotsi leha e le life tse ka 'nang tsa e-ba teng. phenylaminomethyl]-1-methyl-1H-benzimidazol-5-ylcarbonyl]-N-(2-pyridyl)-beta-alanine ethyl ester e na le ts'episo ho k'hemistri ea meriana, lipatlisiso tsa baeloji, le organic synthesis.Leha ho le joalo, lipatlisiso tse ling le liteko lia hlokahala ho bula bokhoni ba eona bo felletseng le ho tseba hore na e sebelisoa joang mafapheng ana.